KN-62是细胞通透性的CaMKⅡ抑制剂，Ki值为0.9 nM，直接与CAMKII的钙调蛋白结合位点相结合，不能抑制其它类的钙调蛋白敏感激酶，也是P2X7受体拮抗剂。据报道，KN-62在高浓度下能抑制GSK3β、PRAK和MAPKAP-K2。
参考文献
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-25~-15℃保存，有效期3年。
