ARRY-380 (HER2-Inhibitor-1; ARRY-380)是一种高效的、选择性的HER2抑制剂，其IC₅₀值为8 nM。

参考文献

[1] Pheneger, T., et al. In vitro and in vivo activity of ARRY-380: A potent, small molecule inhibitor of ErbB2. Presented at the American Association of Cancer Research 100th Annual Meeting Apr 18-22, 2009; Cancer Res 69 (abstr 1795).

[2] Victoria Dinkel, et al. ARRY-380, a potent, small molecule inhibitor of ErbB2, increases survival in intracranial ErbB2+ xenograft models in mice.

冰袋运输。粉末直接保存于-20℃，有效期3年。建议分装后-20℃干燥保存，避免反复冻融。