PF-AKT400是一种有效的ATP竞争性选择性Akt抑制剂，对PKBα（Akt1）具有极高的抑制活性，其选择性是PKA的900倍。

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-25~-15℃避光保存，有效期3年。

[1] Freeman-Cook KD, Autry C, Borzillo G, Gordon D, Barbacci-Tobin E, Bernardo V, Briere D, Clark T, Corbett M, Jakubczak J, Kakar S, Knauth E, Lippa B, Luzzio MJ, Mansour M, Martinelli G, Marx M, Nelson K, Pandit J, Rajamohan F, Robinson S, Subramanyam C, Wei L, Wythes M, Morris J. Design of selective, ATP-competitive inhibitors of Akt. J Med Chem. 2010 Jun 24;53(12):4615-22. doi: 10.1021/jm1003842. Erratum in: J Med Chem. 2010 Aug 12;53(15):5895. PMID: 20481595.