Cisapride
产品介绍
Cisapride是一种口服活性非选择性5-HT4受体激动剂，同时具有hERG通道阻断作用，作为胃促动力剂可显著刺激胃肠运动功能。
产品性质
产品特色
| 英文别名 (English Synonym) | Cisapride |
| 中文名称 (Chinese Name) | 西沙比利 |
| 靶点 (Target) | 5-HT Receptor |
| 通路 (Pathway) | Neuroscience |
| CAS号 (CAS NO.) | 81098-60-4 |
| 分子式 (Formula) | C23H29ClFN3O4 |
| 分子量 (Molecular Weight) | 465.95 |
| 纯度 (Purity) | ≥98% |
| 溶解性 (Solubility) | 溶于DMSO |
存储条件
-25~-15℃保存，有效期3年
COA
已发表文献
[1] Toga T, Kohmura Y, Kawatsu R. The 5-HT(4) agonists cisapride, mosapride, and CJ-033466, a Novel potent compound, exhibit different human ether-a-go-go-related gene (hERG)-blocking activities. J Pharmacol Sci. 2007 Oct;105(2):207-10. doi: 10.1254/jphs.sc0070243. Epub 2007 Oct 6. PMID: 17928736.
[2] Mine Y, Yoshikawa T, Oku S, Nagai R, Yoshida N, Hosoki K. Comparison of effect of mosapride citrate and existing 5-HT4 receptor agonists on gastrointestinal motility in vivo and in vitro. J Pharmacol Exp Ther. 1997 Dec;283(3):1000-8. PMID: 9399969.
相关产品
联系我们
