Bupivacaine HCl是一种NMDA受体抑制剂,可阻断钠通道、L-型钙通道及钾通道;该药物通过与钠通道胞内结构域结合阻断神经细胞钠离子内流,适用于慢性疼痛及心律失常的研究。
| 英文别名 (English Synonym) | Bupivacaine HCl |
| 中文名称 (Chinese Name) | 盐酸布比卡因 |
| 靶点 (Target) | Sodium Channel |
| 通路 (Pathway) | Membrane Transporter/Ion Channel |
| CAS号 (CAS NO.) | 18010-40-7 |
| 分子式 (Formula) | C18H28N2O·HCl |
| 分子量 (Molecular Weight) | 324.89 |
| 纯度 (Purity) | ≥98% |
| 溶解性 (Solubility) | 溶于DMSO |
-25~-15℃保存,有效期3年
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