Vatalanib dihydrochloride 瓦他拉尼二盐酸盐 VEGFR2/KDR抑制剂|CAS 212141-51-0（54600ES）

Vatalanib dihydrochloride，又称瓦他拉尼二盐酸盐，是苯胺邻苯二甲酸衍生物，是可口服的VEGFR2/KDR抑制剂，IC₅₀为37 nM，抑制血管生成。Vatalanib dihydrochloride作用于VEGFR1/FLT1、VEGFR2/Flk1和PDGFRβ的IC₅₀值为77 nM、270 nM和580 nM。

参考文献

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-25~-15℃保存，有效期3年。