Quinacrine hydrochloride hydrate 奎纳克林二盐酸盐二水合物
产品介绍
Quinacrine hydrochloride hydrate(亦称Mepacrine hydrochloride hydrate)兼具抗疟与抗肿瘤活性,其作用机制涉及抑制NF-κB信号通路并激活p53依赖的细胞凋亡途径,从而在体内外模型中有效诱导肿瘤细胞程序性死亡。
产品性质
产品特色
/
存储条件
2~8℃避光保存,有效期3年。
COA
已发表文献
[1] Wu X, Wang Y, Wang H, Wang Q, Wang L, Miao J, Cui F, Wang J. Quinacrine Inhibits Cell Growth and Induces Apoptosis in Human Gastric Cancer Cell Line SGC-7901. Curr Ther Res Clin Exp. 2012 Feb;73(1-2):52-64. doi: 10.1016/j.curtheres.2012.02.003. PMID: 24653512; PMCID: PMC3954015.
[2] Eriksson A, Chantzi E, Fryknäs M, Gullbo J, Nygren P, Gustafsson M, Höglund M, Larsson R. Towards repositioning of quinacrine for treatment of acute myeloid leukemia - Promising synergies and in vivo effects. Leuk Res. 2017 Dec;63:41-46. doi: 10.1016/j.leukres.2017.10.012. Epub 2017 Oct 28. PMID: 29100024.
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