Carprofen,又称卡洛芬、卡布洛芬或卡唑布洛芬,是一种非甾体类抗炎剂,具有抗炎和镇痛的作用,多用作兽药。Carprofen是多靶点FAAH/COX 抑制剂,作用于犬类COX2,IC50为30 nM。卡洛芬对体液免疫和细胞免疫反应也有调节作用。
参考文献
1.Favia AD, et al. Identification and characterization of carprofen as a multitarget fatty acid amide hydrolase/cyclooxygenase inhibitor. J Med Chem. 2012 Oct 25;55(20):8807-26.
2.Waldherr K, et al. In vitro cytoprotective effects of acetylsalicylic acid, carprofen, meloxicam, or robenacoxib against apoptosis induced by sodium nitroprusside in canine cruciate ligament cells. Am J Vet Res. 2012 Nov;73(11):1752-8.
3.Sessions JK, et al. In vivo effects of carprofen, deracoxib, and etodolac on prostanoid production in blood, gastric mucosa, and synovial fluid in dogs with chronic osteoarthritis. Am J Vet Res. 2005 May;66(5):812-7.
冰袋运输。粉末直接保存于-20℃,有效期3年。建议分装后-20℃干燥保存,避免反复冻融。