Icatibant 艾替班特
产品介绍
Icatibant(HOE-140)是强效且特异的缓激肽B2受体拮抗剂,其IC50值为1.07nM,Ki值为0.798nM。
产品性质
产品特色
/
存储条件
-85~-65℃避光保存,有效期2年。
COA
已发表文献
[1] Bawolak MT, Fortin JP, Vogel LK, Adam A, Marceau F. The bradykinin B2 receptor antagonist icatibant (Hoe 140) blocks aminopeptidase N at micromolar concentrations: off-target alterations of signaling mediated by the bradykinin B1 and angiotensin receptors. Eur J Pharmacol. 2006 Dec 3;551(1-3):108-11. doi: 10.1016/j.ejphar.2006.08.077. Epub 2006 Sep 8. PMID: 17026984.[2]Arai Y, Takanashi H, Kitagawa H, Wirth KJ, Okayasu I. Effect of icatibant, a bradykinin B2 receptor antagonist, on the development of experimental ulcerative colitis in mice. Dig Dis Sci. 1999 Apr;44(4):845-51. doi: 10.1023/a:1026694732602. PMID: 10219847.
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