Sarcosine,又称肌氨酸,是一种非蛋白质氨基酸,是竞争性的GlyT1抑制剂,也是NMDAR的协同激动剂,通过增加甘氨酸的浓度增强NMDA受体的功能,具有抗痉挛作用,可用作染料稳定剂,也可以提高人的智力等。
参考文献
[1] Zhang HX, Lyons-Warren A, Thio LL. The glycine transport inhibitor sarcosine is an inhibitory glycine receptor agonist. Neuropharmacology. 2009 Oct-Nov;57(5-6):551-5. doi: 10.1016/j.neuropharm.2009.07.019(IF:4.367).
[2] Chen HH, Stoker A, Markou A, et, al. The glutamatergic compounds sarcosine and N-acetylcysteine ameliorate prepulse inhibition deficits in metabotropic glutamate 5 receptor knockout mice. Psychopharmacology (Berl). 2010 May;209(4):343-50. doi: 10.1007/s00213-010-1802-2(IF:3.424).
[3] Lee MY, Lin YR, Tu YS, et, al. Effects of sarcosine and N, N-dimethylglycine on NMDA receptor-mediated excitatory field potentials. J Biomed Sci. 2017 Feb 28;24(1):18. doi: 10.1186/s12929-016-0314-8(IF:5.203).
-25~-15℃保存,有效期3年。