Rivastigmine Tartrate (ENA 713, SDZ-ENA 713, ENA713),又称酒石酸卡巴拉汀、利斯的明酒石酸盐、卡巴拉汀酒石酸盐、酒石酸利伐斯的明或酒石酸利凡斯的明,是一种可口服的胆碱酯酶抑制剂,IC50为5.5 μM,通过抑制胆碱能神经元对乙酰胆碱的降解而促进胆碱能神经传导,进而促进认知功能,临床上用于治疗阿尔茨海默病。
参考文献
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