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抑制剂激活剂与常用试剂
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Stachydrine 水苏碱
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Stachydrine是益母草的主要活性成分,在促进血液循环、祛除瘀血方面具有传统药用价值。作为一种脯氨酸季铵盐衍生物,它广泛存在于苜蓿属植物中,并可作为尿液中的渗透保护剂。该化合物能够有效抑制NF-κB信号通路。

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存储条件

-25~-15℃避光保存,有效期3年。

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已发表文献

[1] Guo W, Zhang C, Liao YL, Lv R, Wei HC. [Effect of Leonurus stachydrine on myocardial cell hypertrophy]. Zhong Yao Cai. 2012 Jun;35(6):940-3. Chinese. PMID: 23236831.[2]Yin J, Zhang ZW, Yu WJ, Liao JY, Luo XG, Shen YJ. Stachydrine, a major constituent of the Chinese herb leonurus heterophyllus sweet, ameliorates human umbilical vein endothelial cells injury induced by anoxia-reoxygenation. Am J Chin Med. 2010;38(1):157-71. doi: 10.1142/S0192415X10007737. PMID: 20128052.[3]Rathee P, Rathee D, Rathee D, Rathee S. In vitro anticancer activity of stachydrine isolated from Capparis decidua on prostate cancer cell lines. Nat Prod Res. 2012;26(18):1737-40. doi: 10.1080/14786419.2011.608673. Epub 2011 Oct 11. PMID: 21988653.[4]Zhang C, Shan XL, Liao YL, Zhao P, Guo W, Wei HC, Lu R. Effects of stachydrine on norepinephrine-induced neonatal rat cardiac myocytes hypertrophy and intracellular calcium transients. BMC Complement Altern Med. 2014 Dec 8;14:474. doi: 10.1186/1472-6882-14-474. PMID: 25488774; PMCID: PMC4295334.[5]Zhang C, Lu Y, Tong QQ, Zhang L, Guan YF, Wang SJ, Xing ZH. Effect of stachydrine on endoplasmic reticulum stress-induced apoptosis in rat kidney after unilateral ureteral obstruction. J Asian Nat Prod Res. 2013;15(4):373-81. doi: 10.1080/10286020.2013.769964. Epub 2013 Mar 6. PMID: 23464629.

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